SCHEMBL28866735

SCHEMBL28866735

O=CNc1cc(Br)cc2cccnc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.50
KMT2A Q03164 5/20 0.50
BLM P54132 2/20 0.50
CASP3 P42574 1/20 0.50
CASP6 P55212 1/20 0.50
SENP8 Q96LD8 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
TDP1 Q9NUW8 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
APAF1 O14727 2/20 0.41
KDR P35968 2/20 0.41
POLB P06746 1/20 0.41
WDR5 P61964 1/20 0.40
SLC40A1 Q9NP59 5/20 0.39
HTT P42858 2/20 0.39
ALOX15 P16050 1/20 0.39
GLO1 Q04760 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14910896 0.79 MEN1 (0.50) MEN1KMT2ABLMCASP3CASP6
SCHEMBL3425376 0.78 GLO1 (0.56) MEN1KMT2ACASP3SENP8SENP7
SCHEMBL18788338 0.76 CCR1 (0.51) MEN1KMT2ATDP1L3MBTL1SLC40A1
SCHEMBL6589447 0.74 TRIM24 (0.52) MEN1KMT2ATDP1L3MBTL1KDR
SCHEMBL31565225 0.73 TDP1 (0.53) MEN1KMT2ABLMCASP3CASP6
SCHEMBL4466489 0.73 SLC40A1 (0.74) MEN1KMT2ATDP1POLBSLC40A1
SCHEMBL14345508 0.72 SLC40A1 (0.43) MEN1KMT2ATDP1L3MBTL1POLB
SCHEMBL23645096 0.72 TMEM97 (0.46) MEN1KMT2ABLMCASP3CASP6
SCHEMBL416258 0.70 MEN1 (0.73) MEN1KMT2ATDP1POLBSLC40A1
SCHEMBL15961561 0.70 MMP2 (0.56) TDP1HTTALOX15TP53KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884061-A 1,2,4- triazine -3- amine derivant, preparation method and its application in medicine 江苏恒瑞医药股份有限公司 2018-11-23 CN disclosed