SCHEMBL28868541

SCHEMBL28868541

O=C(O)[C@@H]1CCN(Cc2ccnc(Br)c2F)C1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
S1PR1 P21453 8/20 0.44
SYK P43405 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
S1PR5 Q9H228 7/20 0.43
S1PR4 O95977 1/20 0.43
S1PR3 Q99500 1/20 0.43
PDCD1LG2 Q9BQ51 2/20 0.41
CD274 Q9NZQ7 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28868545 1.00 ALDH1A1 (0.44) ALDH1A1S1PR1SYKL3MBTL1S1PR5
SCHEMBL20296352 0.82 CCR5 (0.43) ALDH1A1S1PR1SYKPDCD1LG2CD274
SCHEMBL30740137 0.82 CCR5 (0.43) ALDH1A1S1PR1SYKPDCD1LG2CD274
SCHEMBL20296354 0.82 CCR5 (0.43) ALDH1A1S1PR1SYKPDCD1LG2CD274
SCHEMBL30021389 0.81 CYP2D6 (0.49) ALDH1A1L3MBTL1
SCHEMBL28868539 0.81 ALDH1A1 (0.45) ALDH1A1L3MBTL1CD274
SCHEMBL4664521 0.77 FAAH (0.55) ALDH1A1S1PR1SYKL3MBTL1S1PR5
SCHEMBL4664522 0.77 FAAH (0.55) ALDH1A1S1PR1SYKL3MBTL1S1PR5
SCHEMBL28868640 0.76 CD274 (0.44) SYKPDCD1LG2CD274
SCHEMBL28868653 0.76 CYP1A2 (0.48) CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232109-A PD-1/PD-L1 small molecule inhibitor and application thereof in medicines 广东东阳光药业有限公司 2022-10-25 CN disclosed