SCHEMBL28868640

SCHEMBL28868640

OC1CN(Cc2ccnc(Br)c2F)C1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 11/20 0.44
PDCD1LG2 Q9BQ51 3/20 0.44
PDCD1 Q15116 7/20 0.38
SYK P43405 7/20 0.36
PDE1B Q01064 1/20 0.32
KDR P35968 1/20 0.32
CCR5 P51681 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30740137 0.89 CCR5 (0.43) CD274PDCD1LG2SYKCCR5
SCHEMBL20296354 0.89 CCR5 (0.43) CD274PDCD1LG2SYKCCR5
SCHEMBL20296352 0.89 CCR5 (0.43) CD274PDCD1LG2SYKCCR5
SCHEMBL28957010 0.82 CD274 (0.36) CD274PDCD1LG2PDCD1
SCHEMBL29225552 0.80 ALDH1A1 (0.45)
SCHEMBL28868549 0.77 CD274 (0.35) CD274PDCD1LG2PDCD1
SCHEMBL28868545 0.76 ALDH1A1 (0.44) CD274PDCD1LG2SYK
SCHEMBL28868541 0.76 ALDH1A1 (0.44) CD274PDCD1LG2SYK
SCHEMBL28868539 0.72 ALDH1A1 (0.45) CD274PDCD1
SCHEMBL30021389 0.72 CYP2D6 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232109-A PD-1/PD-L1 small molecule inhibitor and application thereof in medicines 广东东阳光药业有限公司 2022-10-25 CN disclosed