SCHEMBL28868671

SCHEMBL28868671

O=C1CN(Cc2ccnc(Br)c2F)CCN1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
KMT2A Q03164 1/20 0.39
ATM Q13315 1/20 0.39
PDCD1 Q15116 1/20 0.39
CD274 Q9NZQ7 1/20 0.39
SCN9A Q15858 3/20 0.38
GRM2 Q14416 1/20 0.37
POLB P06746 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
FGFR1 P11362 2/20 0.36
NPSR1 Q6W5P4 1/20 0.35
SLC2A1 P11166 2/20 0.35
EGFR P00533 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29225552 0.77 ALDH1A1 (0.45) ALDH1A1KDM4EATMPOLBCYP1A2
SCHEMBL28868663 0.75 CD274 (0.45) PDCD1CD274
SCHEMBL28868624 0.75 CD274 (0.45) PDCD1CD274
SCHEMBL15206491 0.74 KDM5C (0.49) ALDH1A1KDM4EKMT2AATMPDCD1
SCHEMBL22445634 0.71 KDM4E (0.55) ALDH1A1KDM4EKMT2AATMGRM2
SCHEMBL28868640 0.71 CD274 (0.44) PDCD1CD274
SCHEMBL17513334 0.71 SIGMAR1 (0.51) ALDH1A1KDM4EKMT2AATMPOLB
SCHEMBL15206345 0.70 KMT2A (0.40) ALDH1A1KDM4EKMT2AATMPDCD1
SCHEMBL14875655 0.70 AOC1 (0.42) ALDH1A1KDM4EKMT2AATMPDCD1
SCHEMBL1427302 0.70 ALDH1A1 (0.47) ALDH1A1KDM4EKMT2AATMPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232109-A PD-1/PD-L1 small molecule inhibitor and application thereof in medicines 广东东阳光药业有限公司 2022-10-25 CN disclosed