SCHEMBL28869321

SCHEMBL28869321

Cc1[nH]cc([N+](=O)[O-])c1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
TDP1 Q9NUW8 2/20 0.39
HSD17B10 Q99714 1/20 0.38
ERN1 O75460 1/20 0.37
TSHR P16473 5/20 0.36
CYP3A4 P08684 2/20 0.36
GPR35 Q9HC97 1/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ATM Q13315 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RAB9A P51151 1/20 0.35
ALDH1A1 P00352 2/20 0.34
HIF1A Q16665 1/20 0.34
CYP1A2 P05177 1/20 0.33
RECQL P46063 1/20 0.33
ESPL1 Q14674 1/20 0.33
CASP6 P55212 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22576052 0.76 KDM4E (0.55) KDM4ETDP1HSD17B10TSHRCYP3A4
SCHEMBL28479770 0.75 ALDH1A1 (0.40) KDM4ETDP1TSHRCYP3A4MAPT
SCHEMBL9676449 0.69 TDP1 (0.50) KDM4ETDP1HSD17B10TSHRCYP3A4
SCHEMBL5313843 0.68 KDM4E (0.42) KDM4ETDP1HSD17B10ERN1TSHR
SCHEMBL722679 0.68 KDM4E (0.55) KDM4ETDP1HSD17B10TSHRCYP3A4
SCHEMBL1636077 0.67 TDP1 (0.60) KDM4ETDP1HSD17B10TSHRCYP3A4
SCHEMBL19420578 0.67 GPR35 (0.61) KDM4ETDP1HSD17B10TSHRCYP3A4
SCHEMBL1200250 0.67 KDM4E (0.53) KDM4ETDP1HSD17B10TSHRCYP3A4
SCHEMBL9451720 0.67 KDM4E (0.41) KDM4ETDP1HSD17B10TSHRMAPT
SCHEMBL2388710 0.67 TSHR (0.50) KDM4ETDP1TSHRGPR35L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311846-A Novel 6-membered Heteroaromatic Substituted Cyanoindole Derivatives as NIK Inhibitors 杨森制药有限公司 2019-02-05 CN disclosed