SCHEMBL28869801

SCHEMBL28869801

O=C(Cc1ccc2ccccc2c1)Nc1ccc(C(=O)NO)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.69
HDAC1 Q13547 6/20 0.68
HDAC3 O15379 4/20 0.68
HDAC8 Q9BY41 4/20 0.68
HDAC4 P56524 3/20 0.68
HDAC6 Q9UBN7 3/20 0.68
NLRP3 Q96P20 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.59
MEN1 O00255 5/20 0.58
KMT2A Q03164 5/20 0.58
HDAC7 Q8WUI4 2/20 0.58
HDAC2 Q92769 2/20 0.58
HDAC10 Q969S8 1/20 0.58
HDAC11 Q96DB2 1/20 0.58
HDAC9 Q9UKV0 1/20 0.58
HDAC5 Q9UQL6 1/20 0.58
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.56
MAPT P10636 1/20 0.56
HPGD P15428 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29936636 1.00 NR1H4 (0.69) NR1H4HDAC1HDAC3HDAC8HDAC4
SCHEMBL28799744 0.92 NR1H4 (0.61) NR1H4HDAC1HDAC3HDAC8HDAC4
SCHEMBL28869815 0.87 NR1H4 (0.79) NR1H4HDAC1HDAC3HDAC8HDAC4
SCHEMBL28869806 0.87 NLRP3 (0.68) NR1H4HDAC1HDAC3HDAC8HDAC4
SCHEMBL29936235 0.87 NLRP3 (0.68) NR1H4HDAC1HDAC3HDAC8HDAC4
SCHEMBL7311581 0.85 HDAC1 (0.56) NR1H4HDAC1HDAC3HDAC8HDAC4
SCHEMBL9367263 0.84 NR1H4 (0.83) NR1H4HDAC1HDAC3HDAC8HDAC4
SCHEMBL13533414 0.83 NR1H4 (0.76) NR1H4HDAC1HDAC3HDAC8HDAC4
SCHEMBL675578 0.83 KMT2A (0.76) HDAC1HDAC3HDAC8HDAC4HDAC6
SCHEMBL28869822 0.83 RAB9A (0.71) NR1H4HDAC1HDAC3HDAC8HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115093359-B Compound, pharmaceutical composition and application thereof in field of vasodilation or antiviral 山东第一医科大学(山东省医学科学院) 2023-06-09 CN claimed
CN-115093359-A Compound, pharmaceutical composition and application of compound and pharmaceutical composition in field of blood vessel expansion or virus resistance 山东第一医科大学(山东省医学科学院) 2022-09-23 CN claimed
CN-116478070-A Compound, pharmaceutical composition and application thereof in field of vasodilation or antiviral 山东第一医科大学(山东省医学科学院) 2023-07-25 CN disclosed
CN-115093359-B Compound, pharmaceutical composition and application thereof in field of vasodilation or antiviral 山东第一医科大学(山东省医学科学院) 2023-06-09 CN disclosed
CN-115093359-A Compound, pharmaceutical composition and application of compound and pharmaceutical composition in field of blood vessel expansion or virus resistance 山东第一医科大学(山东省医学科学院) 2022-09-23 CN disclosed