SCHEMBL28869822

SCHEMBL28869822

COC(=O)c1ccc(NC(=O)Cc2ccc3ccccc3c2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.71
NPC1 O15118 1/20 0.71
NR1H4 Q96RI1 1/20 0.67
MEN1 O00255 6/20 0.65
KMT2A Q03164 6/20 0.65
MAPK1 P28482 1/20 0.64
ALDH1A1 P00352 5/20 0.62
KDM4E B2RXH2 2/20 0.62
L3MBTL1 Q9Y468 1/20 0.61
MAPK10 P53779 2/20 0.60
MAPK8 P45983 1/20 0.60
NLRP3 Q96P20 1/20 0.59
MAPT P10636 4/20 0.55
LMNA P02545 3/20 0.55
HPGD P15428 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
GSK3A P49840 1/20 0.55
RIOK2 Q9BVS4 1/20 0.55
HDAC3 O15379 1/20 0.54
HDAC4 P56524 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28957115 0.87 MEN1 (0.73) RAB9ANPC1NR1H4MEN1KMT2A
SCHEMBL14344626 0.86 MEN1 (0.76) RAB9ANPC1NR1H4MEN1KMT2A
SCHEMBL13451638 0.86 NR1H4 (0.74) NR1H4MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL28869814 0.85 NR1H4 (0.73) RAB9ANPC1NR1H4MEN1KMT2A
SCHEMBL13451637 0.83 NR1H4 (0.74) RAB9ANPC1NR1H4MEN1KMT2A
SCHEMBL9367263 0.83 NR1H4 (0.83) RAB9ANPC1NR1H4MEN1KMT2A
SCHEMBL29936636 0.83 NR1H4 (0.69) NR1H4MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL28869801 0.83 NR1H4 (0.69) NR1H4MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL13533414 0.82 NR1H4 (0.76) NR1H4MEN1KMT2AALDH1A1KDM4E
SCHEMBL2038480 0.81 L3MBTL1 (0.76) NR1H4MEN1KMT2AALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478070-A Compound, pharmaceutical composition and application thereof in field of vasodilation or antiviral 山东第一医科大学(山东省医学科学院) 2023-07-25 CN disclosed
CN-115093359-B Compound, pharmaceutical composition and application thereof in field of vasodilation or antiviral 山东第一医科大学(山东省医学科学院) 2023-06-09 CN disclosed
CN-115093359-A Compound, pharmaceutical composition and application of compound and pharmaceutical composition in field of blood vessel expansion or virus resistance 山东第一医科大学(山东省医学科学院) 2022-09-23 CN disclosed