SCHEMBL28869893

SCHEMBL28869893

O=c1ccc2ncc(CBr)cc2[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 1/20 0.39
RPS6KA3 P51812 1/20 0.39
CSNK2A1 P68400 1/20 0.39
PLK3 Q9H4B4 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PDE3B Q13370 7/20 0.37
PDE3A Q14432 7/20 0.37
SMYD3 Q9H7B4 1/20 0.36
MAPK1 P28482 1/20 0.35
MAPT P10636 1/20 0.32
HCAR1 Q9BXC0 4/20 0.32
CA12 O43570 2/20 0.32
CA9 Q16790 2/20 0.32
F11 P03951 1/20 0.32
PARP1 P09874 1/20 0.32
CA1 P00915 1/20 0.32
CA3 P07451 1/20 0.32
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32
CA5A P35218 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30011367 1.00 MAPKAPK2 (0.39) MAPKAPK2RPS6KA3CSNK2A1PLK3ALDH1A1
SCHEMBL27752625 0.83 MAPKAPK2 (0.39) MAPKAPK2RPS6KA3CSNK2A1PLK3ALDH1A1
SCHEMBL28869879 0.83 PDE3B (0.44) MAPKAPK2RPS6KA3CSNK2A1PLK3ALDH1A1
SCHEMBL19751457 0.83 PDE3B (0.44) MAPKAPK2RPS6KA3CSNK2A1PLK3ALDH1A1
SCHEMBL30010831 0.83 PDE3B (0.44) MAPKAPK2RPS6KA3CSNK2A1PLK3ALDH1A1
SCHEMBL4135759 0.77 DYRK1A (0.49) MAPKAPK2RPS6KA3CSNK2A1PLK3ALDH1A1
SCHEMBL31093789 0.75 F11 (0.47) MAPKAPK2RPS6KA3CSNK2A1PLK3ALDH1A1
SCHEMBL29115637 0.74 ATAD2 (0.50) PARP1
SCHEMBL29960862 0.74 ATAD2 (0.50) PARP1
SCHEMBL29960664 0.74 PARP1 (0.45) ALDH1A1MAPTPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232121-B Pyridine derivative and application thereof in medicine 成都百裕制药股份有限公司 2023-08-29 CN disclosed
CN-115232121-A Pyridine derivative and application thereof in medicine 成都百裕制药股份有限公司 2022-10-25 CN disclosed