SCHEMBL28871014

SCHEMBL28871014

Brc1ccc(Br)cc1.Nc1cc(F)c(F)cc1N

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
ALOX15 P16050 2/20 0.48
MAPK1 P28482 1/20 0.48
CYP2A6 P11509 1/20 0.44
DGAT1 O75907 1/20 0.40
HTR2A P28223 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
KDM1A O60341 2/20 0.38
KDM1B Q8NB78 1/20 0.38
MAPT P10636 2/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
PTK2 Q05397 1/20 0.37
GLA P06280 1/20 0.37
DPP4 P27487 1/20 0.36
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL102552 0.82 PTK2 (0.54) ALDH1A1ALOX15MAPK1MAPTMEN1
SCHEMBL29363736 0.82 PTK2 (0.54) ALDH1A1ALOX15MAPK1MAPTMEN1
Hydrochloric Acid SCHEMBL10335452 0.78 PTK2 (0.50) ALDH1A1ALOX15MEN1KMT2APTK2
Hydrochloric Acid SCHEMBL10335450 0.78 PTK2 (0.50) ALDH1A1ALOX15MEN1KMT2APTK2
SCHEMBL109380 0.76
SCHEMBL57179 0.76
SCHEMBL29849481 0.76
SCHEMBL2536617 0.74 ALDH1A1 (0.41) ALDH1A1KDM1AKDM1BMAPTMEN1
SCHEMBL241198 0.74 ALDH1A1 (0.42) ALDH1A1KDM1AKDM1BMAPTMEN1
SCHEMBL29902922 0.74 ALDH1A1 (0.42) ALDH1A1KDM1AKDM1BMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113683601-A Diaza-benzo-fluoranthene compound and preparation method and application thereof 广东工业大学 2021-11-23 CN claimed
CN-113683601-B Diaza-benzo-fluoranthene compound and preparation method and application thereof 广东工业大学 2022-09-20 CN disclosed
CN-113683601-A Diaza-benzo-fluoranthene compound and preparation method and application thereof 广东工业大学 2021-11-23 CN disclosed