SCHEMBL28873403

SCHEMBL28873403

CC(C)C1CN(Cl)c2ccccc2C(C2CCCCC2)=N1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.39
CCKBR P32239 13/20 0.36
PTH1R Q03431 4/20 0.35
PTPRC P08575 1/20 0.34
PTPRF P10586 1/20 0.34
PTPN1 P18031 1/20 0.34
CDC25B P30305 1/20 0.34
CCKAR P32238 2/20 0.33
OXTR P30559 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28295463 0.75 GABRA1 (0.43) CHRM1CCKBR
SCHEMBL9008757 0.65 ALDH1A1 (0.42) CCKBRPTH1RCCKAROXTR
SCHEMBL9008759 0.65 ALDH1A1 (0.42) CCKBRPTH1RCCKAROXTR
SCHEMBL9008752 0.65 ALDH1A1 (0.42) CCKBRPTH1RCCKAROXTR
SCHEMBL4414712 0.65 GABRP (0.56) CCKBRCCKAR
SCHEMBL7682526 0.65 GABRP (0.56) CCKBRCCKAR
SCHEMBL8824651 0.65 GABRP (0.56) CCKBRCCKAR
SCHEMBL9383632 0.65 CCKBR (0.37) CCKBRPTH1R
SCHEMBL8824718 0.65 GABRP (0.56) CCKBRCCKAR
SCHEMBL9383622 0.65 CCKBR (0.37) CCKBRPTH1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109906220-A For treating the 1,3- dihydro -1,4- benzodiazepine * -2- thione compounds of CNS related disease 豪夫迈·罗氏有限公司 2019-06-18 CN claimed
CN-109906220-A For treating the 1,3- dihydro -1,4- benzodiazepine * -2- thione compounds of CNS related disease 豪夫迈·罗氏有限公司 2019-06-18 CN disclosed