SCHEMBL28889237

SCHEMBL28889237

CNC(=O)SNC(=O)C(c1ccc(C)cc1)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.39
ACACB O00763 2/20 0.36
SORT1 Q99523 2/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPT P10636 3/20 0.34
KDM4E B2RXH2 1/20 0.34
PSEN1 P49768 3/20 0.33
PSEN2 P49810 3/20 0.33
APH1B Q8WW43 3/20 0.33
NCSTN Q92542 3/20 0.33
APH1A Q96BI3 3/20 0.33
PSENEN Q9NZ42 3/20 0.33
CYP2D6 P10635 2/20 0.33
P2RY1 P47900 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
GPR139 Q6DWJ6 1/20 0.32
SYK P43405 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28889194 0.89 ADRB2 (0.37) ADRB2SORT1ALDH1A1GAAL3MBTL1
SCHEMBL29894640 0.85 HDAC4 (0.40) ADRB2ALDH1A1L3MBTL1MAPTP2RY1
SCHEMBL28889386 0.85 HDAC4 (0.40) ADRB2ALDH1A1L3MBTL1MAPTP2RY1
SCHEMBL28889213 0.84 ADRB2 (0.41) ADRB2ACACBSORT1ALDH1A1GAA
SCHEMBL28889308 0.83 ADRB2 (0.38) ADRB2SORT1ALDH1A1GAAL3MBTL1
SCHEMBL29893753 0.82 ADRB2 (0.37) ADRB2SORT1ALDH1A1GAAL3MBTL1
SCHEMBL28889284 0.82 ADRB2 (0.37) ADRB2SORT1ALDH1A1GAAL3MBTL1
SCHEMBL29942364 0.82 ADRB2 (0.40) ADRB2ACACBSORT1ALDH1A1GAA
SCHEMBL28959159 0.81 ADRB2 (0.38) ADRB2ALDH1A1GAAL3MBTL1MAPT
SCHEMBL28889336 0.81 HDAC4 (0.41) ADRB2ALDH1A1L3MBTL1P2RY1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed