SCHEMBL28889381

SCHEMBL28889381

COc1ncccc1C(C(N)=O)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.39
GPBAR1 Q8TDU6 5/20 0.38
P2RY1 P47900 3/20 0.38
KCNN4 O15554 1/20 0.37
ALDH1A1 P00352 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MAT2A P31153 1/20 0.36
TRPV3 Q8NET8 1/20 0.35
NFE2L2 Q16236 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LRRK2 Q5S007 1/20 0.35
NOS3 P29474 1/20 0.35
NOS2 P35228 1/20 0.35
AHR P35869 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28994016 0.86 ADRB2 (0.40) ADRB2TRPV3
SCHEMBL28889283 0.85 ADRB2 (0.41) ADRB2GPBAR1KCNN4ALDH1A1L3MBTL1
SCHEMBL28889298 0.83 ADRB2 (0.39) ADRB2KCNN4ALDH1A1L3MBTL1TRPV3
SCHEMBL28889349 0.83 P2RY1 (0.41) ADRB2P2RY1ALDH1A1L3MBTL1
SCHEMBL28889159 0.82 GPBAR1 (0.41) ADRB2GPBAR1ALDH1A1L3MBTL1
SCHEMBL28889339 0.82 ADRB2 (0.42) ADRB2KCNN4ALDH1A1L3MBTL1TRPV3
SCHEMBL28889277 0.81 P2RY1 (0.38) ADRB2GPBAR1P2RY1KCNN4ALDH1A1
SCHEMBL28889367 0.81 ADRB2 (0.41) ADRB2KCNN4ALDH1A1L3MBTL1TRPV3
SCHEMBL28959168 0.80 HDAC4 (0.44) ADRB2P2RY1TRPV3NOS3NOS2
SCHEMBL28889221 0.79 ADRB2 (0.41) ADRB2ALDH1A1L3MBTL1TRPV3NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed