SCHEMBL28889277

SCHEMBL28889277

CNC(=S)NC(=O)C(c1cc(C(F)(F)F)ccn1)c1cccnc1OC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY1 P47900 8/20 0.38
ADRB2 P07550 1/20 0.36
KCNN4 O15554 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.34
KDR P35968 1/20 0.34
CLK2 P49760 1/20 0.34
IRAK1 P51617 1/20 0.34
NEK4 P51957 1/20 0.34
MAP4K2 Q12851 1/20 0.34
HIPK4 Q8NE63 1/20 0.34
SRPK1 Q96SB4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28889238 0.91 ADRB2 (0.37) P2RY1ADRB2LMNAPOLBCYP3A4
SCHEMBL29893632 0.91 ADRB2 (0.37) P2RY1ADRB2LMNAPOLBCYP3A4
SCHEMBL28889349 0.90 P2RY1 (0.41) P2RY1ADRB2LMNAPOLBCYP3A4
SCHEMBL29942209 0.87 ADRB2 (0.38) P2RY1ADRB2KCNN4LMNAPOLB
SCHEMBL29941794 0.84 ADRB2 (0.38) ADRB2KCNN4LMNAPOLBALDH1A1
SCHEMBL29942331 0.84 ADRB2 (0.38) P2RY1ADRB2KCNN4LMNAPOLB
SCHEMBL29941803 0.84 HDAC4 (0.42) P2RY1ADRB2LMNAPOLBALDH1A1
SCHEMBL29941823 0.83 ADRB2 (0.40) ADRB2LMNAPOLBALDH1A1L3MBTL1
SCHEMBL28889381 0.81 ADRB2 (0.39) P2RY1ADRB2KCNN4ALDH1A1L3MBTL1
SCHEMBL28889196 0.81 TACR1 (0.43) ADRB2LMNAALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed