SCHEMBL28894423

SCHEMBL28894423

CC(C)(C)NC(=O)c1cnn(C/C(=C\F)COC(N)=O)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 4/20 0.44
MAOB P27338 1/20 0.44
JAK2 O60674 1/20 0.33
ACHE P22303 1/20 0.32
LMNA P02545 2/20 0.32
CYP2C19 P33261 2/20 0.32
GAA P10253 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
KDR P35968 3/20 0.32
MAPT P10636 1/20 0.31
GFER P55789 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KLKB1 P03952 3/20 0.31
KLK1 P06870 1/20 0.31
ROCK1 Q13464 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28894427 1.00 AOC3 (0.44) AOC3MAOBJAK2ACHELMNA
SCHEMBL28432378 0.88 KLKB1 (0.34) AOC3MAOBACHELMNACYP2C19
SCHEMBL28432376 0.88 KLKB1 (0.34) AOC3MAOBACHELMNACYP2C19
SCHEMBL28426244 0.86 LMNA (0.37) LMNACYP2C19MAPTGFERNPSR1
SCHEMBL28426245 0.86 LMNA (0.37) LMNACYP2C19MAPTGFERNPSR1
SCHEMBL22216397 0.85 AOC3 (0.51) AOC3MAOBJAK2ACHELMNA
SCHEMBL22216190 0.85 AOC3 (0.42) AOC3MAOBACHELMNACYP2C19
SCHEMBL23907239 0.84 AOC3 (0.36) AOC3MAOBACHELMNACYP2C19
SCHEMBL22216189 0.82 AOC3 (0.40) AOC3MAOBACHELMNACYP2C19
SCHEMBL28429087 0.82 LOXL2 (0.33) AOC3MAOBACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111434662-B Haloallylamine compound and application thereof 药捷安康(南京)科技股份有限公司 2023-01-10 CN disclosed
CN-111434662-A Haloallylamine compound and application thereof 南京药捷安康生物科技有限公司 2020-07-21 CN disclosed