SCHEMBL22216397

SCHEMBL22216397

CC(C)(C)NC(=O)c1cnn(C/C(=C/F)CN)c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 6/20 0.51
MAOB P27338 1/20 0.51
KLKB1 P03952 5/20 0.35
ACHE P22303 2/20 0.35
LMNA P02545 2/20 0.34
MAPT P10636 1/20 0.34
CYP2C19 P33261 1/20 0.34
GFER P55789 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
JAK2 O60674 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KLK1 P06870 1/20 0.33
HPGD P15428 1/20 0.33
SYK P43405 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22216190 0.90 AOC3 (0.42) AOC3MAOBACHELMNAMAPT
SCHEMBL22216189 0.87 AOC3 (0.40) AOC3MAOBKLKB1ACHELMNA
SCHEMBL22216335 0.86 KLKB1 (0.37) AOC3MAOBKLKB1ACHELMNA
SCHEMBL28894423 0.85 AOC3 (0.44) AOC3MAOBKLKB1ACHELMNA
SCHEMBL28894427 0.85 AOC3 (0.44) AOC3MAOBKLKB1ACHELMNA
SCHEMBL23907200 0.85 AOC3 (0.38) AOC3MAOBKLKB1ACHELMNA
SCHEMBL23907203 0.85 AOC3 (0.38) AOC3MAOBKLKB1ACHELMNA
SCHEMBL22216339 0.84 KLKB1 (0.41) KLKB1LMNAMAPTCYP2C19GFER
SCHEMBL23920660 0.82 L3MBTL1 (0.38) AOC3MAOBKLKB1ACHEL3MBTL1
SCHEMBL28435846 0.81 AOC3 (0.38) AOC3MAOBKLKB1ACHELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111434662-B Haloallylamine compound and application thereof 药捷安康(南京)科技股份有限公司 2023-01-10 CN disclosed
EP-3892621-A1 HALOALLYLAMINE COMPOUNDS AND APPLICATION THEREOF Nanjing Transthera Biosciences Co., Ltd. (CN) 2021-10-13 EP disclosed
WO-2020143763-A1 HALOALLYLAMINE COMPOUNDS AND APPLICATION THEREOF 南京药捷安康生物科技有限公司 2020-07-16 WO disclosed