SCHEMBL28895114

SCHEMBL28895114

COC(=O)c1c(F)cc(NC(=O)OC(C)(C)C)cc1CBr

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.36
AAK1 Q2M2I8 3/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP17A1 P05093 1/20 0.35
ATR Q13535 1/20 0.35
BDKRB1 P46663 1/20 0.35
MAPT P10636 1/20 0.35
EGLN2 Q96KS0 2/20 0.34
SYK P43405 1/20 0.34
RORC P51449 4/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA9 Q16790 1/20 0.34
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
LEF1 Q9UJU2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16137967 0.87 MAPT (0.41) ENPP2KDM4ECYP17A1ATRMAPT
SCHEMBL28895294 0.86 RORC (0.35) ENPP2AAK1KDM4ECYP17A1ATR
SCHEMBL28895279 0.82 CA12 (0.41) ENPP2KDM4ECYP17A1ATRMAPT
SCHEMBL793197 0.81 ATR (0.42) ENPP2ATRMAPTEGLN2SYK
SCHEMBL22941793 0.79 CA12 (0.44) AAK1CYP17A1SYKRORCCA12
SCHEMBL22941851 0.78 CA12 (0.41) AAK1KDM4ECYP17A1SYKRORC
SCHEMBL28895200 0.78 SYK (0.36) ENPP2KDM4ECYP17A1ATRMAPT
SCHEMBL13928829 0.77 CYP17A1 (0.36) AAK1CYP17A1EGLN2SYKCA12
SCHEMBL12931081 0.77 CYP17A1 (0.36) ENPP2AAK1KDM4ECYP17A1RORC
SCHEMBL17629762 0.77 RARA (0.43) CYP17A1EGLN2SYKRORCCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114315805-A Aromatic ring-fused cyclic lactone thiohydantoin compound and preparation method and application thereof 中国科学院上海药物研究所 2022-04-12 CN disclosed