SCHEMBL28895200

SCHEMBL28895200

C=Cc1cc(NC(=O)OC(C)(C)C)cc(F)c1C(=O)OC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.36
ATR Q13535 1/20 0.35
MAPT P10636 1/20 0.35
EGLN2 Q96KS0 2/20 0.34
F13A1 P00488 1/20 0.34
TGM2 P21980 1/20 0.34
TGM1 P22735 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA9 Q16790 1/20 0.34
NAMPT P43490 1/20 0.34
MAP4K4 O95819 1/20 0.34
ENPP2 Q13822 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
ACVR1B P36896 1/20 0.33
TGFBR1 P36897 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16137967 0.87 MAPT (0.41) SYKATRMAPTEGLN2CA12
SCHEMBL28895279 0.82 CA12 (0.41) SYKATRMAPTEGLN2CA12
SCHEMBL793197 0.81 ATR (0.42) SYKATRMAPTEGLN2CA12
SCHEMBL28895114 0.78 ENPP2 (0.36) SYKATRMAPTEGLN2CA12
SCHEMBL19511536 0.77 ATR (0.44) ATRCA12CA1CA9NAMPT
SCHEMBL17629762 0.77 RARA (0.43) SYKEGLN2CA12CA1CA9
SCHEMBL28895294 0.77 RORC (0.35) SYKATRMAPTEGLN2CA12
SCHEMBL17643122 0.76 CA12 (0.39) SYKEGLN2CA12CA1CA9
SCHEMBL28895142 0.75 CA12 (0.41) SYKEGLN2F13A1TGM2TGM1
SCHEMBL15076456 0.75 CA12 (0.42) SYKEGLN2CA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114315805-A Aromatic ring-fused cyclic lactone thiohydantoin compound and preparation method and application thereof 中国科学院上海药物研究所 2022-04-12 CN disclosed