SCHEMBL28895294

SCHEMBL28895294

COC(=O)c1c(F)cc(NC(=O)OC(C)(C)C)cc1CCO

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP17A1 P05093 1/20 0.34
ATR Q13535 1/20 0.34
MAPT P10636 1/20 0.34
EGLN2 Q96KS0 2/20 0.34
SYK P43405 1/20 0.34
ENPP2 Q13822 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA9 Q16790 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
NPC1 O15118 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28895114 0.86 ENPP2 (0.36) RORCKDM4ECYP17A1ATRMAPT
SCHEMBL16137967 0.86 MAPT (0.41) KDM4ECYP17A1ATRMAPTEGLN2
SCHEMBL28895279 0.81 CA12 (0.41) RORCKDM4ECYP17A1ATRMAPT
SCHEMBL793197 0.80 ATR (0.42) RORCATRMAPTEGLN2SYK
SCHEMBL19511628 0.78 ATR (0.43) CYP17A1ATRCA12CA1CA9
SCHEMBL15076460 0.77 CA12 (0.40) RORCCYP17A1EGLN2SYKCA12
SCHEMBL28895200 0.77 SYK (0.36) RORCKDM4ECYP17A1ATRMAPT
SCHEMBL17629762 0.76 RARA (0.43) RORCCYP17A1EGLN2SYKCA12
SCHEMBL17643122 0.74 CA12 (0.39) RORCCYP17A1EGLN2SYKCA12
SCHEMBL15076459 0.74 CA12 (0.40) RORCCYP17A1EGLN2SYKCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114315805-A Aromatic ring-fused cyclic lactone thiohydantoin compound and preparation method and application thereof 中国科学院上海药物研究所 2022-04-12 CN disclosed