SCHEMBL28895380

SCHEMBL28895380

[CH2]C(N(c1ccc(N)cc1)S(C)(=O)=O)C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.37
CYP3A4 P08684 4/20 0.35
TDP1 Q9NUW8 3/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPK1 P28482 2/20 0.35
TP53 P04637 1/20 0.35
ALOX15 P16050 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.33
TSHR P16473 3/20 0.32
PSMD14 O00487 1/20 0.32
RECQL P46063 1/20 0.32
GFER P55789 1/20 0.32
LMNA P02545 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MPO P05164 1/20 0.31
CYP2C9 P11712 1/20 0.31
HTR6 P50406 1/20 0.31
CA12 O43570 3/20 0.31
CA1 P00915 3/20 0.31
CA2 P00918 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2993431 0.78 ALDH1A1 (0.43) HSD11B1CYP3A4TDP1ALDH1A1MAPK1
SCHEMBL11296691 0.70 ALDH1A1 (0.36) HSD11B1CYP3A4TDP1ALDH1A1MAPK1
SCHEMBL3030207 0.68 TDP1 (0.48) CYP3A4TDP1ALDH1A1MAPK1TP53
SCHEMBL1916178 0.66 ALDH1A1 (0.52) CYP3A4TDP1ALDH1A1MAPK1TP53
SCHEMBL28547556 0.65 TSHR (0.41) CYP3A4TDP1ALDH1A1MAPK1TP53
SCHEMBL7850305 0.64 MMP2 (0.39) CYP3A4TDP1ALDH1A1MAPK1TP53
SCHEMBL4241968 0.62 SMN1; SMN2 (0.39) CYP3A4TDP1ALDH1A1MAPK1TP53
SCHEMBL20389164 0.61 ESR1 (0.61) HSD11B1CYP3A4TDP1ALDH1A1L3MBTL1
SCHEMBL2991577 0.60 CYP3A4 (0.39) HSD11B1CYP3A4TDP1ALDH1A1MAPK1
SCHEMBL5109986 0.60 PSIP1 (0.44) KDM4ECA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115052663-A ALK5 inhibitor conjugates and uses thereof 辛瑟斯治疗股份有限公司 2022-09-13 CN disclosed