SCHEMBL28898024

SCHEMBL28898024

CCOc1cc(OC(N)=O)ncc1Br

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NCOA1 Q15788 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
TSHR P16473 3/20 0.43
HSD17B10 Q99714 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.40
LMNA P02545 3/20 0.39
HTT P42858 1/20 0.39
MAPK1 P28482 2/20 0.37
MAPT P10636 1/20 0.36
POLB P06746 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
NPC1 O15118 1/20 0.36
CYP3A4 P08684 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28898026 0.88 SMN1; SMN2 (0.43) NCOA1NCOA3HSD17B10KMT2AMEN1
SCHEMBL21830618 0.78 NNMT (0.47) NCOA1NCOA3TSHRKMT2AMEN1
SCHEMBL15881230 0.78 NNMT (0.46) TSHRHSD17B10KMT2AMEN1ALDH1A1
SCHEMBL23089103 0.75 NNMT (0.31) KMT2AMEN1
SCHEMBL28876608 0.74 ALDH1A1 (0.35) TSHRKMT2AMEN1ALDH1A1MAPT
SCHEMBL9572460 0.73 MEN1 (0.36) KMT2AMEN1MKNK1MKNK2
SCHEMBL17559336 0.73 TSHR (0.54) NCOA1NCOA3TSHRHSD17B10KMT2A
SCHEMBL23089282 0.72 GRM4 (0.35) HSD17B10KMT2AMEN1ALDH1A1HTT
SCHEMBL15527772 0.72 LMNA (0.41) NCOA1NCOA3TSHRHSD17B10KMT2A
SCHEMBL28912500 0.71 PLAU (0.33) KMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111527078-B Pyridinecarbonyl derivatives and their therapeutic use as TRPC6 inhibitors 勃林格殷格翰国际公司 2023-06-02 CN disclosed
CN-111527078-A Pyridinecarbonyl derivatives and their therapeutic use as TRPC6 inhibitors 勃林格殷格翰国际公司 2020-08-11 CN disclosed