SCHEMBL28899220

SCHEMBL28899220

COc1ccc(Cn2cc(Br)c3ccc(NCC(=O)C4CC4)cc3c2=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.43
NPC1 O15118 2/20 0.43
TSHR P16473 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
TP53 P04637 1/20 0.43
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
NFKB1 P19838 1/20 0.43
HTT P42858 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
BRD4 O60885 1/20 0.43
KDM4E B2RXH2 3/20 0.41
ATM Q13315 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAPK10 P53779 3/20 0.40
ALDH1A1 P00352 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30095522 1.00 LMNA (0.43) LMNANPC1TSHRRAB9ASMN1; SMN2
SCHEMBL30095463 0.80 BRD4 (0.40) LMNANPC1TSHRRAB9ASMN1; SMN2
SCHEMBL28899157 0.80 BRD4 (0.40) LMNANPC1TSHRRAB9ASMN1; SMN2
SCHEMBL28899155 0.77 RAB9A (0.48) LMNANPC1TSHRRAB9ASMN1; SMN2
SCHEMBL28899159 0.74 MAPT (0.44) LMNATP53MAPK10ALDH1A1HDAC1
SCHEMBL30095433 0.74 MAPT (0.44) LMNATP53MAPK10ALDH1A1HDAC1
SCHEMBL28321534 0.72 HDAC3 (0.62) TSHRTP53POLBHTTALDH1A1
SCHEMBL14915956 0.68 MAPK8 (0.52) LMNATSHRTP53ALDH1A1MAPT
SCHEMBL15010499 0.67 MAPK8 (0.47) LMNATP53HDAC1HDAC2HDAC6
SCHEMBL19679824 0.66 MAPK10 (0.52) LMNATP53BRD4KDM4EMAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109456308-B Heterocyclic compounds as ASK inhibitors and their use 南京圣和药业股份有限公司 2022-11-29 CN disclosed
CN-109456308-A Heterocyclic compound and its application as ASK inhibitor 南京圣和药业股份有限公司 2019-03-12 CN disclosed