SCHEMBL28899155

SCHEMBL28899155

COc1ccc(Cn2ncc3ccc(NCC(=O)C4CC4)cc3c2=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.48
NPC1 O15118 3/20 0.48
TSHR P16473 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
LMNA P02545 2/20 0.48
HPGD P15428 2/20 0.48
TP53 P04637 1/20 0.48
POLB P06746 1/20 0.48
NFKB1 P19838 1/20 0.48
HTT P42858 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
KDM4E B2RXH2 2/20 0.45
HSD17B10 Q99714 2/20 0.45
ATM Q13315 1/20 0.45
NPBWR1 P48145 7/20 0.45
AURKA O14965 1/20 0.43
GRK2 P25098 1/20 0.43
ROCK1 Q13464 1/20 0.43
RPS6KA1 Q15418 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30095522 0.77 LMNA (0.43) RAB9ANPC1TSHRSMN1; SMN2LMNA
SCHEMBL28899220 0.77 LMNA (0.43) RAB9ANPC1TSHRSMN1; SMN2LMNA
SCHEMBL28899162 0.76 NPBWR1 (0.56) HTTHSD17B10NPBWR1AURKAGRK2
SCHEMBL28321534 0.74 HDAC3 (0.62) TSHRTP53POLBHTTMTNR1A
SCHEMBL30579886 0.72 TDP1 (0.64) RAB9ANPC1HTTHSD17B10NPBWR1
SCHEMBL28899217 0.72 MAPT (0.52) SMN1; SMN2NPBWR1AURKAGRK2ROCK1
SCHEMBL28899175 0.70 MAP3K5 (0.48) NPBWR1AURKAGRK2ROCK1RPS6KA1
SCHEMBL28899197 0.70 AURKA (0.43) NPBWR1AURKAGRK2ROCK1RPS6KA1
SCHEMBL22226011 0.69 NPBWR1 (0.62) TP53NPBWR1AURKAGRK2ROCK1
SCHEMBL25432622 0.69 NPBWR1 (0.55) NPBWR1PKMPKLRPDE1APDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109456308-B Heterocyclic compounds as ASK inhibitors and their use 南京圣和药业股份有限公司 2022-11-29 CN disclosed
CN-109456308-A Heterocyclic compound and its application as ASK inhibitor 南京圣和药业股份有限公司 2019-03-12 CN disclosed