SCHEMBL28906367

SCHEMBL28906367

Fc1cccc(-c2[nH]c3ccccc3c2Cc2c(-c3cccc(F)c3)[nH]c3ccccc23)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.64
HTR2C P28335 5/20 0.64
DRD2 P14416 3/20 0.64
LMNA P02545 1/20 0.54
HPGD P15428 1/20 0.54
CNR1 P21554 3/20 0.50
SIRT1 Q96EB6 1/20 0.49
TDO2 P48775 1/20 0.49
TUBB4A P04350 3/20 0.48
TUBB P07437 3/20 0.48
TUBA3C P0DPH7 3/20 0.48
TUBA1B P68363 3/20 0.48
TUBA4A P68366 3/20 0.48
TUBB4B P68371 3/20 0.48
TUBB3 Q13509 3/20 0.48
TUBB2A Q13885 3/20 0.48
TUBB8 Q3ZCM7 3/20 0.48
TUBA3E Q6PEY2 3/20 0.48
TUBA1A Q71U36 3/20 0.48
TUBA1C Q9BQE3 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30046753 1.00 HTR2A (0.64) HTR2AHTR2CDRD2LMNAHPGD
SCHEMBL28906353 0.81 HTR2A (0.61) HTR2AHTR2CDRD2HPGDCNR1
SCHEMBL28906516 0.81 HTR2A (0.62) HTR2AHTR2CDRD2CNR1TUBB4A
SCHEMBL28906409 0.81 HTR6 (0.65) HTR2AHTR2CDRD2CNR1TDO2
SCHEMBL30047360 0.81 HTR6 (0.65) HTR2AHTR2CDRD2CNR1TDO2
SCHEMBL28906384 0.81 NR1I3 (0.51) HTR2AHTR2CDRD2HPGDSIRT1
SCHEMBL28906432 0.81 FNTA (0.51) HTR2AHTR2CDRD2CNR1TDO2
SCHEMBL30047453 0.81 NR1I3 (0.51) HTR2AHTR2CDRD2HPGDSIRT1
SCHEMBL28906368 0.81 KDM4E (0.51) HTR2AHTR2CLMNAHPGDCNR1
SCHEMBL28906422 0.81 LMNA (0.51) HTR2AHTR2CDRD2LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304533-B Bisindolemethane type alpha-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2024-04-12 CN disclosed
CN-117567447-A Thiophene-containing bis-indolomethane type a-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2024-02-20 CN disclosed
CN-115304533-A Bis-indole methane type alpha-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2022-11-08 CN disclosed