SCHEMBL28906371

SCHEMBL28906371

Clc1ccc(-c2[nH]c3ccccc3c2Cc2c(-c3ccc(Cl)cc3)[nH]c3ccccc23)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.61
HTR2C P28335 2/20 0.61
DRD2 P14416 1/20 0.61
CCNB2 O95067 2/20 0.57
CDK1 P06493 2/20 0.57
CCNB1 P14635 2/20 0.57
CCNB3 Q8WWL7 2/20 0.57
MAPT P10636 3/20 0.55
KDM4E B2RXH2 2/20 0.55
PTGS2 P35354 2/20 0.49
KMT2A Q03164 2/20 0.49
PDE10A Q9Y233 1/20 0.49
GSK3A P49840 1/20 0.48
GSK3B P49841 1/20 0.48
PRNP P04156 1/20 0.48
TUBB4A P04350 3/20 0.47
TUBB P07437 3/20 0.47
TUBA3C P0DPH7 3/20 0.47
TUBA1B P68363 3/20 0.47
TUBA4A P68366 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7495375 0.93 HTR2A (0.58) HTR2AHTR2CDRD2CCNB2CDK1
SCHEMBL6992348 0.88 TUBB4A (0.57) HTR2AHTR2CDRD2CCNB2CDK1
SCHEMBL6990745 0.86 DRD2 (0.52) HTR2AHTR2CDRD2CCNB2CDK1
SCHEMBL28906516 0.85 HTR2A (0.62) HTR2AHTR2CDRD2TUBB4ATUBB
SCHEMBL14074161 0.83 HTR2A (0.63) HTR2AHTR2CDRD2CCNB2CDK1
SCHEMBL11495770 0.82 HTR2A (0.65) HTR2AHTR2CDRD2CCNB2CDK1
SCHEMBL28906353 0.82 HTR2A (0.61) HTR2AHTR2CDRD2MAPTKDM4E
SCHEMBL28906377 0.82 PTGS2 (0.49) HTR2AHTR2CDRD2MAPTPTGS2
SCHEMBL28906369 0.82 MAPT (0.55) HTR2AHTR2CDRD2MAPTPTGS2
SCHEMBL28906438 0.81 TUBB4A (0.67) MAPTKDM4EPTGS2KMT2APDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304533-B Bisindolemethane type alpha-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2024-04-12 CN disclosed
CN-117567447-A Thiophene-containing bis-indolomethane type a-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2024-02-20 CN disclosed
CN-115304533-A Bis-indole methane type alpha-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2022-11-08 CN disclosed