SCHEMBL28906383

SCHEMBL28906383

Cc1ccc2c(N(C)c3c(-c4ccccc4)[nH]c4cc(C)ccc34)c(-c3ccccc3)[nH]c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.54
HPGD P15428 4/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
MDM4 O15151 1/20 0.48
MDM2 Q00987 1/20 0.48
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 2/20 0.44
GFER P55789 2/20 0.44
CNR1 P21554 3/20 0.43
PTGS2 P35354 2/20 0.43
HSD17B10 Q99714 3/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28906358 0.83 ESR1 (0.57) KDM4EALDH1A1PTGS2HSD17B10HTR2A
SCHEMBL28906378 0.83 TUBB4A (0.53) HPGDALDH1A1CNR1PTGS2HTR2A
SCHEMBL28024124 0.80 ESR1 (0.65) KIF11HPGDCYP1A2CYP2D6CYP2C9
SCHEMBL28960401 0.77 MDM4 (0.68) KIF11HPGDCYP1A2CYP2D6CYP2C9
SCHEMBL28486502 0.75 KIF11 (0.51) KIF11HPGDCYP1A2CYP2D6CYP2C9
SCHEMBL28906355 0.73 PTGS2 (0.53) HPGDKDM4EALDH1A1CNR1PTGS2
SCHEMBL28855249 0.73 KIF11 (0.49) KIF11HPGDCYP1A2CYP2D6CYP2C9
SCHEMBL19256986 0.73 KIF11 (0.67) KIF11HPGDMDM4MDM2KDM4E
SCHEMBL12939133 0.71 F2 (0.61) KIF11HPGDCYP1A2CYP2D6CYP2C9
SCHEMBL607346 0.71 KIF11 (1.00) KIF11KDM4EALDH1A1HSD17B10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304533-A Bis-indole methane type alpha-glucosidase inhibitor and preparation method and application thereof 中国医学科学院药用植物研究所云南分所 2022-11-08 CN disclosed