SCHEMBL28907136

SCHEMBL28907136

COC(C)=Cc1c([N+](=O)[O-])ccc(Oc2ccnc3cc(OCc4ccccc4)c(OC)cc23)c1F

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MET P08581 16/20 0.48
KDR P35968 4/20 0.45
PDGFRA P16234 1/20 0.45
AXL P30530 2/20 0.44
MST1R Q04912 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28530276 0.93 MET (0.45) METKDRPDGFRAAXLMST1R
SCHEMBL28512289 0.85 MET (0.47) METKDRPDGFRAAXLMST1R
SCHEMBL1549776 0.84 MET (0.48) METKDRPDGFRAAXLMST1R
SCHEMBL2335546 0.83 KDR (0.49) METKDRPDGFRAAXLMST1R
SCHEMBL28447507 0.82 CTSV (0.45)
SCHEMBL1549363 0.80 MET (0.43) METKDRPDGFRAAXLMST1R
SCHEMBL10296341 0.80 MET (0.42) METKDRPDGFRAAXLMST1R
SCHEMBL1876626 0.79 AXL (0.54) METKDRPDGFRAAXL
SCHEMBL371803 0.78 MET (0.55) METKDRPDGFRAAXLMST1R
SCHEMBL4483017 0.78 MET (0.55) METKDRPDGFRAAXLMST1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110357856-B Arotinib hydrochloride intermediate and preparation method of Arotinib hydrochloride 新发药业有限公司 2021-02-26 CN disclosed