SCHEMBL28920185

SCHEMBL28920185

CC(C)n1ncc2cc([N+](=O)[O-])cc(Br)c21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.38
ALDH1A1 P00352 4/20 0.38
CYP3A4 P08684 1/20 0.38
ESPL1 Q14674 1/20 0.35
GLS O94925 1/20 0.35
GLA P06280 1/20 0.34
TSHR P16473 1/20 0.33
MAPT P10636 2/20 0.33
CRHBP P24387 1/20 0.33
HTT P42858 1/20 0.33
CRHR2 Q13324 1/20 0.33
CREBBP Q92793 1/20 0.33
POLB P06746 1/20 0.32
MAOB P27338 1/20 0.32
NOS1 P29475 1/20 0.32
FLT3 P36888 1/20 0.32
CYP19A1 P11511 1/20 0.32
HSP90AA1 P07900 2/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31662360 0.82 ALDH1A1 (0.40) NQO2ALDH1A1CYP3A4ESPL1GLS
SCHEMBL28920240 0.78 RAB9A (0.44) NQO2ALDH1A1CYP3A4ESPL1GLS
SCHEMBL29730504 0.76 ALDH1A1 (0.44) ALDH1A1GLSMAPTHTTPOLB
SCHEMBL31304574 0.75 GLS (0.55) ALDH1A1CYP3A4GLSTSHRMAPT
SCHEMBL5352816 0.75 GLS (0.55) ALDH1A1CYP3A4GLSTSHRMAPT
SCHEMBL28920149 0.73 GAA (0.34) MAPTCHEK1DAPK3LIMK1
SCHEMBL29534076 0.72 KMT2A (0.38) ALDH1A1CYP3A4GLSTSHRMAPT
SCHEMBL22939501 0.72 KDM4E (0.42) TSHRPOLBKMT2A
SCHEMBL31510404 0.72 GLS (0.45) ALDH1A1CYP3A4GLSTSHRMAPT
SCHEMBL2144733 0.72 GLS (0.45) ALDH1A1CYP3A4GLSTSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115490709-A KRASG12D inhibitor and application thereof in medicine 四川海思科制药有限公司 2022-12-20 CN disclosed