SCHEMBL28920149

SCHEMBL28920149

CC(C)n1ncc2cc(N)cc(Br)c21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
CHEK1 O14757 1/20 0.31
AURKA O14965 1/20 0.31
DAPK3 O43293 1/20 0.31
CSNK1A1 P48729 1/20 0.31
GSK3A P49840 1/20 0.31
LIMK1 P53667 1/20 0.31
IKBKE Q14164 1/20 0.31
MAPK14 Q16539 1/20 0.31
TAOK1 Q7L7X3 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
DYRK1B Q9Y463 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
ADORA1 P30542 1/20 0.31
PIK3CD O00329 1/20 0.31
ABL1 P00519 1/20 0.31
EGFR P00533 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15910568 0.81 SYK (0.38) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL28920192 0.75 HASPIN (0.48) GAAMAPTCHEK1AURKADAPK3
SCHEMBL22939501 0.74 KDM4E (0.42) ADORA3ADORA2AADORA2BADORA1KDM4E
SCHEMBL4083412 0.74 NOS1 (0.34) BACE1MAPK1
SCHEMBL28920185 0.73 NQO2 (0.38) MAPTCHEK1DAPK3LIMK1
SCHEMBL19762454 0.72 PDE1B (0.36) KDM4E
SCHEMBL22939496 0.71 ALDH1A1 (0.41) GAAMAPTADORA3ADORA2AADORA2B
SCHEMBL15910720 0.70 SYK (0.33) KDM4EMAPK1
SCHEMBL3353513 0.70 ADORA3 (0.41) AURKAADORA3ADORA2AADORA2BADORA1
SCHEMBL31304384 0.70 ADORA3 (0.41) AURKAADORA3ADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115490709-A KRASG12D inhibitor and application thereof in medicine 四川海思科制药有限公司 2022-12-20 CN disclosed