SCHEMBL28940976

SCHEMBL28940976

CNC(=O)c1ncc(NC(=O)O)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HTM Q9NXG6 2/20 0.41
SMN1; SMN2 Q16637 4/20 0.39
RAB9A P51151 5/20 0.38
NPC1 O15118 3/20 0.38
CNR1 P21554 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
BAZ2B Q9UIF8 1/20 0.37
SORT1 Q99523 1/20 0.36
KCNQ3 O43525 2/20 0.36
KCNQ2 O43526 2/20 0.36
MAPT P10636 1/20 0.35
KDM4E B2RXH2 2/20 0.35
MITF O75030 1/20 0.35
XBP1 P17861 1/20 0.35
PAX8 Q06710 1/20 0.35
KLF5 Q13887 1/20 0.35
KMT2A Q03164 1/20 0.35
KCNE1 P15382 1/20 0.35
KCNQ1 P51787 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12179242 0.79 CNR1 (0.42) SMN1; SMN2RAB9ANPC1CNR1BAZ2B
SCHEMBL459529 0.77 P4HTM (0.42) P4HTMSMN1; SMN2RAB9ANPC1ALDH1A1
SCHEMBL22227949 0.77 P4HTM (0.55) P4HTMSMN1; SMN2RAB9ANPC1ALDH1A1
SCHEMBL24756311 0.76 ALDH1A1 (0.54) SMN1; SMN2RAB9AALDH1A1GAAMAPT
SCHEMBL28940905 0.76 P4HTM (0.36) P4HTMSMN1; SMN2RAB9ANPC1ALDH1A1
SCHEMBL28941020 0.76 HDAC1 (0.37) P4HTMSMN1; SMN2RAB9ANPC1ALDH1A1
SCHEMBL28940972 0.75 CNR1 (0.43) P4HTMRAB9ANPC1CNR1ALDH1A1
SCHEMBL28940920 0.75 ACR (0.40) P4HTMSMN1; SMN2ALDH1A1KDM4EKMT2A
SCHEMBL28940979 0.75 CNR2 (0.38) P4HTMSMN1; SMN2RAB9ANPC1ALDH1A1
SCHEMBL25738793 0.74 PLK1 (0.50) SMN1; SMN2RAB9ANPC1BAZ2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed