SCHEMBL28940972

SCHEMBL28940972

O=C(O)Nc1cnc(C(=O)NCCO)nc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.43
MMP13 P45452 1/20 0.39
OPRM1 P35372 1/20 0.37
OPRL1 P41146 1/20 0.37
MEN1 O00255 1/20 0.36
CACNA1B Q00975 1/20 0.36
APBA1 Q02410 1/20 0.36
KMT2A Q03164 1/20 0.36
TP53 P04637 1/20 0.36
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALPL P05186 1/20 0.35
P4HTM Q9NXG6 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19145297 0.82 CNR1 (0.51) CNR1MMP13OPRM1OPRL1MEN1
SCHEMBL21379406 0.81 NAMPT (0.48) CNR1P4HTMGCGRMAOB
SCHEMBL21379396 0.80 P4HTM (0.36) CNR1KDM4EALDH1A1POLBP4HTM
SCHEMBL15228258 0.77 KDM4E (0.42) CNR1OPRM1OPRL1MEN1KMT2A
SCHEMBL28940920 0.76 ACR (0.40) MEN1KMT2AKDM4EALDH1A1P4HTM
SCHEMBL28940979 0.76 CNR2 (0.38) ALDH1A1P4HTMNPC1RAB9AGAA
SCHEMBL28940976 0.75 P4HTM (0.41) CNR1KMT2AKDM4EALDH1A1P4HTM
SCHEMBL19105518 0.73 RAB9A (0.47) CNR1MMP13OPRM1OPRL1POLB
SCHEMBL28292622 0.73 ANO1 (0.45) CNR1KMT2APOLB
SCHEMBL22341930 0.73 P2RX7 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed