SCHEMBL28949574

SCHEMBL28949574

OB(O)c1cccc(C(F)F)c1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRB3 P13945 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
FAAH O00519 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
GABRA1 P14867 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
GABRB1 P18505 1/20 0.32
GABRG2 P18507 1/20 0.32
PTGS1 P23219 1/20 0.32
SLC6A2 P23975 1/20 0.32
HTR2C P28335 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29524794 1.00 ENPP2 (0.33) ENPP2ADRB1ADRA2AADRB3ADRA2B
SCHEMBL29951757 0.80 ENPP2 (0.41) ENPP2FAAHCA1CA2LMNA
SCHEMBL4013443 0.80 ENPP2 (0.41) ENPP2FAAHCA1CA2LMNA
SCHEMBL25745449 0.79 ENPP2 (0.42) ENPP2
SCHEMBL29955624 0.78 MAPT (0.33) ENPP2FAAHCA1CA2LMNA
SCHEMBL29956604 0.76 CYP1A2 (0.32) ENPP2FAAHCA1CA2LMNA
SCHEMBL4384 0.73 CES2 (0.43) ENPP2HPGDCES2CES1
SCHEMBL29399046 0.73 CES2 (0.43) ENPP2HPGDCES2CES1
SCHEMBL28971466 0.72 GABRA1 (0.38) ADRB1ADRA2AADRB3ADRA2BADRA2C
SCHEMBL22905245 0.71 GABRA1 (0.46) FAAHCA1CA2LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed