Cyclopropane

Cyclopropane

SCHEMBL28956243

C1CC1.CN(C(=O)c1ccc(N)cc1)c1ccc(CN)cc1

nearest known ligand 0.47

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.47
EGFR P00533 1/20 0.46
ERBB2 P04626 1/20 0.46
LOXL2 Q9Y4K0 2/20 0.44
HIF1A Q16665 1/20 0.43
EPAS1 Q99814 1/20 0.43
MAOA P21397 1/20 0.42
CYP26B1 Q9NR63 1/20 0.41
HTT P42858 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
PPIB P23284 2/20 0.39
KLKB1 P03952 1/20 0.39
MLNR O43193 1/20 0.38
NAMPT P43490 1/20 0.38
TRPV1 Q8NER1 1/20 0.37
PHLPP2 Q6ZVD8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8581201 0.84 KMT2A (0.50) NR1H4EGFRERBB2MAOAHTT
SCHEMBL2127770 0.84 KMT2A (0.50) NR1H4EGFRERBB2MAOAHTT
Cyclopropane SCHEMBL28215074 0.82 LOXL2 (0.54) NR1H4EGFRERBB2LOXL2HTT
SCHEMBL7046909 0.81 KMT2A (0.54) NR1H4EGFRERBB2MAOAHTT
SCHEMBL12812295 0.79 KDM4E (0.59) NR1H4EGFRERBB2LOXL2MAOA
SCHEMBL13973193 0.78 TRPV1 (0.56) NR1H4KDM4ETRPV1
SCHEMBL7406735 0.78 HSD17B1 (0.50) NR1H4EGFRERBB2MAOAHTT
SCHEMBL1749595 0.77 MCHR1 (0.50) EGFRERBB2HIF1AMAOAHTT
SCHEMBL7410067 0.76 CHEK2 (0.49) NR1H4EGFRERBB2MAOAHTT
SCHEMBL7373511 0.76 KMT2A (0.64) EGFRERBB2MAOAHTTHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026039-A New carbocyclic compound as ROR gamma modulators 格兰马克药品股份有限公司 2018-05-11 CN disclosed