SCHEMBL28956705

SCHEMBL28956705

Cc1nc2[nH]c(=O)n(COCC(C)C)c(=O)c2[nH]1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.39
PDE1A P54750 1/20 0.39
PDE1B Q01064 1/20 0.39
PDE1C Q14123 1/20 0.39
ADORA2B P29275 13/20 0.38
ADORA3 P0DMS8 5/20 0.38
ADORA2A P29274 2/20 0.36
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL150604 0.81 PDE1A (0.54) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL14142760 0.71 ADORA2B (0.57) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL387340 0.68 ADORA2B (0.55) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL6381402 0.66 ADORA2B (0.36) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL9031176 0.66 ADORA2B (0.44) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL6033611 0.65 ADORA2B (0.52) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL10535020 0.65 ADORA2B (0.47) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL516430 0.62 PDE2A (0.44) PDE2APDE1APDE1BPDE1CADORA2B
Acetic Acid SCHEMBL28746161 0.62 ADORA2B (0.52) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL6363706 0.61 ADORA1 (0.48) ADORA2BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108699028-A It is substituted 4- phenylpyridine compounds as non-systemic TGR5 agonists 阿德利克斯公司 2018-10-23 CN disclosed