SCHEMBL28958210

SCHEMBL28958210

COC(=O)CNCc1ccccc1.Cc1ccc(S(=O)(=O)O)cc1

nearest known ligand 0.50

Known targets — ChEMBL curated mechanism

ABL1BMXBRAFBTKCHRNA4CHRNB2CSNK1EEGFRERBB2F10FLT1FLT3FLT4IGF1RINSRITKJAK3KDRKITOPRM1PARP1PARP2PDGFRBPIK3CDRAF1RETSLC18A2TECTXKdacAdacBdacCftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.50
CYP1A2 P05177 2/20 0.50
CA12 O43570 2/20 0.50
CA9 Q16790 2/20 0.50
CYP3A4 P08684 1/20 0.50
ATM Q13315 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
MAPT P10636 2/20 0.48
SMN1; SMN2 Q16637 3/20 0.46
LMNA P02545 3/20 0.45
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 2/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
CYP2C9 P11712 1/20 0.43
PKM P14618 1/20 0.42
TP53 P04637 1/20 0.42
GAA P10253 2/20 0.42
HPGD P15428 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4200394 0.88 CA12 (0.54) KMT2ACYP1A2CA12CA9CYP3A4
SCHEMBL29803178 0.83 CA12 (0.58) KMT2ACYP1A2CA12CA9CYP3A4
SCHEMBL717052 0.83 MEN1 (0.50) KMT2AATML3MBTL1MAPTSMN1; SMN2
SCHEMBL19401273 0.83 MEN1 (0.50) KMT2AATML3MBTL1MAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL2840965 0.81 MEN1 (0.49) KMT2ACYP3A4ATMMAPTSMN1; SMN2
SCHEMBL6811685 0.81 KMT2A (0.50) KMT2AATMSMN1; SMN2LMNAALDH1A1
SCHEMBL13731468 0.80 MAPT (0.52) KMT2ACYP1A2CA12CA9CYP3A4
N-Benzylmethylamine SCHEMBL20239926 0.79 CYP3A4 (0.59) KMT2ACYP1A2CA12CA9CYP3A4
SCHEMBL28338890 0.77 L3MBTL1 (0.58) KMT2ACYP1A2CA12CA9CYP3A4
SCHEMBL11624179 0.77 LMNA (0.53) KMT2AMAPTLMNAALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115583903-B Method for rapidly preparing racecadotril 湖北广辰药业有限公司 2024-05-28 CN disclosed
CN-115583903-A Method for rapidly preparing racecadotril 湖北广辰药业有限公司 2023-01-10 CN disclosed