SCHEMBL28964103

SCHEMBL28964103

COc1cc(NC(O)COC(N)=O)c(C(N)=O)cc1OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
KDM4E B2RXH2 1/20 0.47
CYP1A2 P05177 1/20 0.47
SMPD1 P17405 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
CTSV O60911 3/20 0.45
CTSL P07711 3/20 0.45
HTT P42858 1/20 0.44
SRD5A1 P18405 1/20 0.43
SRD5A2 P31213 1/20 0.43
F2 P00734 2/20 0.43
F10 P00742 2/20 0.43
PRSS1 P07477 2/20 0.43
F7 P08709 2/20 0.43
PRSS2 P07478 1/20 0.43
F3 P13726 1/20 0.43
PRSS3 P35030 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19983333 0.81 SMPD1 (0.54) LMNASMN1; SMN2KDM4ESMPD1HDAC1
SCHEMBL874091 0.75 HTT (0.55) LMNASMN1; SMN2KDM4ESMPD1HDAC1
SCHEMBL159448 0.75 HTT (0.55) LMNASMN1; SMN2KDM4ESMPD1HDAC1
SCHEMBL1656948 0.74 SMPD1 (0.53) LMNASMN1; SMN2KDM4ESMPD1HDAC1
SCHEMBL7048751 0.74 SMPD1 (0.53) LMNASMN1; SMN2KDM4ESMPD1HDAC1
SCHEMBL30211021 0.73 CTSV (0.60) SMN1; SMN2KDM4ECYP1A2SMPD1HDAC1
SCHEMBL8039259 0.71 LMNA (0.51) LMNASMN1; SMN2SMPD1HDAC1HDAC8
SCHEMBL23459152 0.71 KDM4E (0.52) SMN1; SMN2KDM4ESMPD1HDAC1HDAC8
SCHEMBL2089698 0.71 KDM4E (0.52) SMN1; SMN2KDM4ESMPD1HDAC1HDAC8
SCHEMBL873729 0.70 MEN1 (0.57) LMNAKDM4ESMPD1HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115677701-A Benzo heterocyclic compound and preparation method and application thereof 昆药集团股份有限公司 2023-02-03 CN disclosed