SCHEMBL8039259

SCHEMBL8039259

COc1cc(C(F)(F)F)c(C(N)=O)cc1OCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.51
HTT P42858 1/20 0.51
SMPD1 P17405 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
NPC1 O15118 1/20 0.48
HPGD P15428 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MRGPRX4 Q96LA9 3/20 0.47
SRD5A1 P18405 2/20 0.47
SRD5A2 P31213 2/20 0.47
RXRA P19793 2/20 0.47
RXRB P28702 1/20 0.47
RXRG P48443 1/20 0.47
CTSV O60911 2/20 0.46
CTSL P07711 2/20 0.46
ATM Q13315 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8035471 0.90 CTSV (0.54) SMPD1HDAC1HDAC8HDAC6NPC1
SCHEMBL8037062 0.86 SMPD1 (0.51) LMNAHTTSMPD1HDAC1HDAC8
SCHEMBL8034962 0.84 HPGD (0.58) LMNAHTTSMPD1HDAC1HDAC8
SCHEMBL24983699 0.83 RXRA (0.58) MRGPRX4RXRARXRBRXRG
SCHEMBL30892446 0.83 RXRA (0.58) MRGPRX4RXRARXRBRXRG
SCHEMBL874091 0.82 HTT (0.55) LMNAHTTSMPD1HDAC1HDAC8
SCHEMBL159448 0.82 HTT (0.55) LMNAHTTSMPD1HDAC1HDAC8
SCHEMBL8023147 0.82 APP (0.46) SMPD1HDAC1HDAC8HDAC6NPC1
SCHEMBL8039263 0.82 SMN1; SMN2 (0.54) LMNAHTTSMPD1HDAC1HDAC8
SCHEMBL8039245 0.82 MRGPRX4 (0.49) LMNAHTTSMPD1HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed