SCHEMBL28973017

SCHEMBL28973017

CC(=O)Nc1cc([N+](=O)[O-])c(Br)nc1OC(F)C(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.44
LMNA P02545 3/20 0.44
NPSR1 Q6W5P4 2/20 0.44
GALR2 O43603 1/20 0.44
MITF O75030 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HSP90AA1 P07900 1/20 0.44
HPGD P15428 1/20 0.44
XBP1 P17861 1/20 0.44
CCR6 P51684 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MAPT P10636 2/20 0.38
KMT2A Q03164 4/20 0.37
HTT P42858 2/20 0.36
SLC9A1 P19634 1/20 0.36
MEN1 O00255 3/20 0.36
GAA P10253 2/20 0.35
EGFR P00533 1/20 0.34
PKM P14618 2/20 0.33
PDE7A Q13946 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28359193 0.91 POLB (0.45) POLBLMNANPSR1GALR2MITF
SCHEMBL28496822 0.86 POLB (0.44) POLBLMNANPSR1GALR2MITF
SCHEMBL24251661 0.83 ALDH1A1 (0.46) POLBLMNANPSR1GALR2MITF
SCHEMBL29756268 0.83 ALDH1A1 (0.46) POLBLMNANPSR1GALR2MITF
SCHEMBL28973016 0.78 MAPT (0.39) POLBLMNANPSR1GALR2MITF
SCHEMBL29389430 0.78 NPSR1 (0.46) POLBLMNANPSR1GALR2MITF
SCHEMBL24251729 0.78 NPSR1 (0.46) POLBLMNANPSR1GALR2MITF
SCHEMBL28359039 0.76 NPSR1 (0.45) POLBLMNANPSR1GALR2MITF
SCHEMBL28973026 0.74 CA1 (0.38) POLBALDH1A1HPGDSMN1; SMN2MAPT
SCHEMBL17490481 0.72 NPSR1 (0.43) POLBLMNANPSR1GALR2MITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115701429-B 4- (1H-indol-1-yl) pyrimidine-2-amino derivative, and preparation method and application thereof 上海和誉生物医药科技有限公司 2024-03-12 CN disclosed
CN-115836064-A Triazine derivative with EGFR (epidermal growth factor receptor) inhibitory activity and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-03-21 CN disclosed
CN-115701429-A 4- (1H-indole-1-yl) pyrimidine-2-amino derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-02-10 CN disclosed