SCHEMBL29756268

SCHEMBL29756268

COc1nc(Br)c([N+](=O)[O-])cc1NC(C)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
NPSR1 Q6W5P4 2/20 0.46
POLB P06746 2/20 0.46
GALR2 O43603 1/20 0.46
MITF O75030 1/20 0.46
LMNA P02545 1/20 0.46
HSP90AA1 P07900 1/20 0.46
HPGD P15428 1/20 0.46
XBP1 P17861 1/20 0.46
CCR6 P51684 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MAPT P10636 4/20 0.43
KMT2A Q03164 5/20 0.41
HTT P42858 2/20 0.41
SLC9A1 P19634 1/20 0.40
PKM P14618 2/20 0.39
GAA P10253 1/20 0.39
MEN1 O00255 3/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24251661 1.00 ALDH1A1 (0.46) ALDH1A1NPSR1POLBGALR2MITF
SCHEMBL10745494 0.87 POLB (0.49) ALDH1A1NPSR1POLBGALR2MITF
SCHEMBL28359193 0.85 POLB (0.45) ALDH1A1NPSR1POLBGALR2MITF
SCHEMBL17490464 0.84 NPSR1 (0.46) ALDH1A1NPSR1POLBGALR2MITF
SCHEMBL28973017 0.83 POLB (0.44) ALDH1A1NPSR1POLBGALR2MITF
SCHEMBL29389430 0.82 NPSR1 (0.46) ALDH1A1NPSR1POLBGALR2MITF
SCHEMBL24251729 0.82 NPSR1 (0.46) ALDH1A1NPSR1POLBGALR2MITF
SCHEMBL31149365 0.80 ALDH1A1 (0.45) ALDH1A1LMNASMN1; SMN2KMT2AHTT
SCHEMBL24251673 0.78 ALDH1A1 (0.44) ALDH1A1NPSR1POLBGALR2MITF
SCHEMBL17490478 0.76 ALDH1A1 (0.42) ALDH1A1NPSR1POLBGALR2MITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115836064-B Triazine derivative with EGFR (epidermal growth factor receptor) inhibition activity as well as preparation method and application thereof 上海和誉生物医药科技有限公司 2024-08-27 CN disclosed
CN-117440945-A Pyrimidine or pyridine derivative, preparation method thereof and application thereof in pharmacy 上海和誉生物医药科技有限公司 2024-01-23 CN disclosed
CN-115867539-A 2, 3-dihydro-1H-pyrrolo [3,2-b ] pyridine derivatives, preparation method and application thereof 上海和誉生物医药科技有限公司 2023-03-28 CN disclosed
CN-115836064-A Triazine derivative with EGFR (epidermal growth factor receptor) inhibitory activity and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-03-21 CN disclosed
CN-110642838-B EGFR inhibitor and preparation and application thereof 江苏威凯尔医药科技有限公司 2022-08-09 CN disclosed
CN-110642836-B EGFR inhibitor and preparation and application thereof 江苏威凯尔医药科技有限公司 2022-08-09 CN disclosed