SCHEMBL24251729

SCHEMBL24251729

CC(=O)Nc1cc([N+](=O)[O-])c(Br)nc1OCC(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.46
ALDH1A1 P00352 3/20 0.46
LMNA P02545 2/20 0.46
GALR2 O43603 1/20 0.46
MITF O75030 1/20 0.46
POLB P06746 1/20 0.46
HSP90AA1 P07900 1/20 0.46
HPGD P15428 1/20 0.46
XBP1 P17861 1/20 0.46
CCR6 P51684 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
AR P10275 2/20 0.40
KMT2A Q03164 3/20 0.39
CNR2 P34972 1/20 0.39
MAPT P10636 3/20 0.38
THRB P10828 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29389430 1.00 NPSR1 (0.46) NPSR1ALDH1A1LMNAGALR2MITF
SCHEMBL17490379 0.86 NPSR1 (0.46) NPSR1ALDH1A1LMNAGALR2MITF
SCHEMBL29756268 0.82 ALDH1A1 (0.46) NPSR1ALDH1A1LMNAGALR2MITF
SCHEMBL24251661 0.82 ALDH1A1 (0.46) NPSR1ALDH1A1LMNAGALR2MITF
SCHEMBL24251711 0.81 ALDH1A1 (0.41) NPSR1ALDH1A1LMNAGALR2MITF
SCHEMBL18978915 0.80 ALDH1A1 (0.40) NPSR1ALDH1A1LMNAGALR2MITF
SCHEMBL28359193 0.80 POLB (0.45) NPSR1ALDH1A1LMNAGALR2MITF
SCHEMBL28510516 0.79 ALDH1A1 (0.44) NPSR1ALDH1A1LMNAGALR2MITF
SCHEMBL28973017 0.78 POLB (0.44) NPSR1ALDH1A1LMNAGALR2MITF
SCHEMBL29133283 0.75 WDR5 (0.40) NPSR1ALDH1A1LMNAGALR2MITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115701429-B 4- (1H-indol-1-yl) pyrimidine-2-amino derivative, and preparation method and application thereof 上海和誉生物医药科技有限公司 2024-03-12 CN disclosed
CN-115836064-A Triazine derivative with EGFR (epidermal growth factor receptor) inhibitory activity and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-03-21 CN disclosed
CN-115701429-A 4- (1H-indole-1-yl) pyrimidine-2-amino derivative and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-02-10 CN disclosed
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed