SCHEMBL28985329

SCHEMBL28985329

COc1cc(B(O)O)cc(OC)c1OC.Nc1nc2cccc(Br)n2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 1/20 0.45
NUDT1 P36639 3/20 0.41
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
TUBB2A Q13885 1/20 0.38
TUBB8 Q3ZCM7 1/20 0.38
TUBA3E Q6PEY2 1/20 0.38
TUBA1A Q71U36 1/20 0.38
TUBA1C Q9BQE3 1/20 0.38
TUBB6 Q9BUF5 1/20 0.38
TUBB2B Q9BVA1 1/20 0.38
TUBB1 Q9H4B7 1/20 0.38
AHR P35869 1/20 0.36
EGLN2 Q96KS0 1/20 0.35
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30263737 0.78 JAK1 (0.65) JAK1NUDT1TUBB4ATUBBTUBA3C
SCHEMBL45713 0.76 NUDT1 (0.56) JAK1NUDT1AHREGLN2
SCHEMBL24433 0.70 CYP3A4 (0.56) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL14888861 0.68 JAK1 (0.66) JAK1NUDT1EGLN2MAPTHSP90AB1
SCHEMBL30263741 0.67 JAK2 (0.64) JAK1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL14721848 0.65 CYP3A4 (0.50) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL30263697 0.65 TUBB4A (0.50) JAK1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL2640360 0.65 JAK2 (0.56) JAK1NUDT1EGLN2MAPTJAK2
SCHEMBL3304801 0.64 JAK1 (0.75) JAK1NUDT1EGLN2MAPTJAK2
SCHEMBL7435094 0.63 CYP3A4 (0.42) TUBB4ATUBBTUBA3CTUBA1BTUBA4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115819425-A Triazolo hexa-nitrogen heterocyclic-2-amine compound and preparation method and application thereof 五邑大学 2023-03-21 CN disclosed