SCHEMBL28987252

SCHEMBL28987252

Brc1cnc2cnn(C3CC3)c2c1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.35
DYRK1A Q13627 2/20 0.34
PDE4D Q08499 2/20 0.33
PIK3CD O00329 1/20 0.32
OPRK1 P41145 5/20 0.32
HTR3A P46098 2/20 0.31
KCNH2 Q12809 1/20 0.31
HRH4 Q9H3N8 4/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
KDM1A O60341 1/20 0.30
PDE1A P54750 1/20 0.30
PDE1B Q01064 1/20 0.30
PDE1C Q14123 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28987256 0.93 OPRK1 (0.36) HSD17B10DYRK1AOPRK1HRH4
SCHEMBL25389131 0.76 RXRA (0.43) OPRK1KMT2A
SCHEMBL31104405 0.74 KMO (0.43) PIK3CD
SCHEMBL16595822 0.74 KMO (0.43) PIK3CD
SCHEMBL27402945 0.74 HDAC8 (0.38) HSD17B10PIK3CDOPRK1HTR3AKCNH2
SCHEMBL30853275 0.74 HDAC8 (0.38) HSD17B10PIK3CDOPRK1HTR3AKCNH2
SCHEMBL16302863 0.73 HSD17B10 (0.39) HSD17B10DYRK1AHTTKMT2A
SCHEMBL16913940 0.72 PIK3C3 (0.49) HSD17B10DYRK1A
SCHEMBL15333094 0.72 HSD17B10 (0.46) HSD17B10DYRK1AHRH4HTTKMT2A
SCHEMBL29377303 0.72 HSD17B10 (0.46) HSD17B10DYRK1AHRH4HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116003408-A Heterocyclic compound, and preparation method and application thereof 绵阳市中心医院 2023-04-25 CN disclosed