SCHEMBL28987256

SCHEMBL28987256

Brc1cnc2cnn(C3CCCC3)c2c1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 13/20 0.36
PDE9A O76083 2/20 0.36
HRH4 Q9H3N8 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HCAR3 P49019 1/20 0.33
DYRK1A Q13627 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28987252 0.93 HSD17B10 (0.35) OPRK1HRH4HSD17B10DYRK1A
SCHEMBL25389131 0.79 RXRA (0.43) OPRK1
SCHEMBL2980987 0.75 PIK3CD (0.41) PDE9A
SCHEMBL19698021 0.74 PIK3CD (0.41) PDE9A
SCHEMBL19966455 0.74 KDM5A (0.47) PDE9A
SCHEMBL17677989 0.72 PIK3CD (0.41) PDE9A
SCHEMBL25045382 0.72 HTR7 (0.39) PDE9AHCAR3
SCHEMBL10124057 0.72 ALDH1A1 (0.40) OPRK1PDE9AHSD17B10HCAR3
SCHEMBL24268689 0.71 HCAR3 (0.42) PDE9AHSD17B10HCAR3
SCHEMBL24268646 0.71 NR3C1 (0.39) PDE9AHCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116003408-A Heterocyclic compound, and preparation method and application thereof 绵阳市中心医院 2023-04-25 CN disclosed