SCHEMBL28987465

SCHEMBL28987465

COc1ccc2c(-n3cc4c(n3)CCN(C(=O)O)C4)ccnc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 2/20 0.41
CYP8B1 Q9UNU6 1/20 0.40
PDK2 Q15119 1/20 0.40
GAA P10253 1/20 0.39
PTGS1 P23219 1/20 0.38
CYP2C19 P33261 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
MAPK7 Q13164 1/20 0.38
LMNA P02545 1/20 0.38
KCNH2 Q12809 1/20 0.38
GRM4 Q14833 1/20 0.38
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
NCF1 P14598 1/20 0.37
MET P08581 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPK1 P28482 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24008962 0.88 MAPT (0.48) CYP8B1PDK2GAAMAPK7ESR2
SCHEMBL24008960 0.81 GAA (0.38) CYP8B1GAAKCNH2GRM4NCF1
SCHEMBL3070215 0.79 DHFR (0.46) PTGDR2NCF1
SCHEMBL17202416 0.78 PDK2 (0.52) HSP90AB1PDK2ESR1ESR2
SCHEMBL24008963 0.77 NCF1 (0.45) GAALMNAKCNH2GRM4NCF1
SCHEMBL20303278 0.73 PDK2 (0.43) HSP90AB1PDK2LMNAKCNH2KDM4E
SCHEMBL4069676 0.72 SLC6A9 (0.52) PDK2KCNH2
SCHEMBL3741308 0.71 NCF1 (0.47) GAALMNAKCNH2GRM4NCF1
SCHEMBL4067477 0.70 PDK2 (0.47) HSP90AB1PDK2KCNH2
SCHEMBL3073912 0.69 NCF1 (0.56) GAALMNAKCNH2NCF1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996912-A Iminothiolanone inhibitors of ENPP1 沃拉斯查疗法公司 2023-04-21 CN disclosed