SCHEMBL289883

SCHEMBL289883

N#CC(CNC(=O)C1(NC(=O)O)CCOCC1)c1ccc(I)cc1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSL P07711 10/20 0.37
CTSB P07858 10/20 0.37
CTSS P25774 9/20 0.37
CTSK P43235 2/20 0.37
CTSC P53634 2/20 0.36
KCNH2 Q12809 1/20 0.34
LTB4R Q15722 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.34
TACR2 P21452 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290024 0.86 CTSC (0.49) CTSLCTSBCTSSCTSKCTSC
SCHEMBL288986 0.86 MMP1 (0.41) CTSLCTSBCTSSCTSKCTSC
SCHEMBL290246 0.84 ALDH1A1 (0.41) CTSLCTSBCTSSCTSKCTSC
SCHEMBL290154 0.84 FFAR1 (0.40) CTSLCTSBCTSSCTSKCTSC
SCHEMBL290266 0.82 CTSC (0.38) CTSLCTSBCTSSCTSKCTSC
SCHEMBL289590 0.82 CTSC (0.38) CTSLCTSBCTSSCTSKCTSC
SCHEMBL290312 0.81 CTSC (0.41) CTSLCTSBCTSSCTSKCTSC
SCHEMBL290666 0.81 CTSC (0.38) CTSLCTSBCTSSCTSKCTSC
SCHEMBL290432 0.80 CTSL (0.46) CTSLCTSBCTSS
SCHEMBL289804 0.79 CTSC (0.42) CTSLCTSBCTSSCTSKCTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed