SCHEMBL289905

SCHEMBL289905

CCNC(=O)c1sc(-c2ccc(-c3cc4ccccc4s3)s2)nc1C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.60
NPC1 O15118 3/20 0.60
SMN1; SMN2 Q16637 4/20 0.45
GAA P10253 5/20 0.45
KDM4E B2RXH2 5/20 0.45
ALDH1A1 P00352 5/20 0.44
MAPT P10636 3/20 0.44
NPSR1 Q6W5P4 1/20 0.43
RAB9A P51151 4/20 0.43
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
ESR1 P03372 1/20 0.42
POLB P06746 1/20 0.42
JMJD7 P0C870 1/20 0.42
STAT3 P40763 1/20 0.42
STAT1 P42224 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290238 0.83 SMN1; SMN2 (0.56) HPGDNPC1SMN1; SMN2GAAKDM4E
SCHEMBL288852 0.83 KDM4E (0.59) HPGDNPC1SMN1; SMN2GAAKDM4E
SCHEMBL2787018 0.81 SMN1; SMN2 (0.41) HPGDNPC1SMN1; SMN2GAAKDM4E
SCHEMBL290307 0.81 CD274 (0.61) HPGDSMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL298961 0.77 NPC1 (0.62) HPGDNPC1SMN1; SMN2GAAKDM4E
SCHEMBL289671 0.77 HTR2C (0.57) NPC1SMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL289881 0.76 SMN1; SMN2 (0.61) HPGDNPC1SMN1; SMN2GAAKDM4E
SCHEMBL289614 0.75 KDM4E (0.64) HPGDNPC1SMN1; SMN2GAAKDM4E
SCHEMBL290239 0.75 CYP2A6 (0.42)
SCHEMBL3828069 0.74 LMNA (0.51) HPGDSMN1; SMN2GAAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed