SCHEMBL290239

SCHEMBL290239

Cc1nc(-c2ccc(-c3cc4ccccc4s3)s2)sc1CO

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.42
APP P05067 2/20 0.39
ADRB2 P07550 1/20 0.36
HSD17B1 P14061 1/20 0.36
HSD17B2 P37059 1/20 0.36
CYP19A1 P11511 1/20 0.36
TNIK Q9UKE5 3/20 0.35
STK17B O94768 2/20 0.35
STK17A Q9UEE5 2/20 0.35
CAMKK1 Q8N5S9 1/20 0.35
AURKB Q96GD4 1/20 0.35
CAMKK2 Q96RR4 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
TRPV3 Q8NET8 1/20 0.35
HIPK4 Q8NE63 1/20 0.34
IKBKB O14920 1/20 0.34
LMNA P02545 1/20 0.34
JAK2 O60674 1/20 0.33
JAK3 P52333 1/20 0.33
IDH1 O75874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3822637 0.81 CYP2A6 (0.46) CYP2A6APPADRB2HSD17B1HSD17B2
SCHEMBL288852 0.78 KDM4E (0.59) LMNAJAK2JAK3
SCHEMBL290238 0.78 SMN1; SMN2 (0.56)
SCHEMBL289837 0.77 DPP4 (0.53) LMNA
SCHEMBL3828017 0.77 ALDH1A1 (0.37) TRPV3LMNA
SCHEMBL2787018 0.76 SMN1; SMN2 (0.41) APPSTK17BSTK17ACAMKK1AURKB
SCHEMBL26500221 0.75 APP (0.45) CYP2A6APPHSD17B1HSD17B2CYP19A1
SCHEMBL289905 0.75 HPGD (0.60)
SCHEMBL290100 0.75 CYP2A6 (0.40) CYP2A6APPADRB2HSD17B1HSD17B2
SCHEMBL5148513 0.74 APP (0.57) CYP2A6APPADRB2HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed