SCHEMBL289916

SCHEMBL289916

CCOC(=O)c1sc(-c2ccc(C(=O)c3cccs3)s2)nc1C

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.71
ALDH1A1 P00352 6/20 0.71
RAB9A P51151 6/20 0.58
SMN1; SMN2 Q16637 6/20 0.58
NPC1 O15118 5/20 0.58
HPGD P15428 5/20 0.58
CDC7 O00311 5/20 0.54
DBF4 Q9UBU7 5/20 0.54
LMNA P02545 2/20 0.51
GAA P10253 2/20 0.49
MEN1 O00255 2/20 0.49
TP53 P04637 2/20 0.49
CASP1 P29466 2/20 0.49
KMT2A Q03164 2/20 0.49
HSD17B10 Q99714 2/20 0.49
NFKB1 P19838 2/20 0.49
NFKB2 Q00653 2/20 0.49
RELA Q04206 2/20 0.49
POLB P06746 1/20 0.49
MAPK1 P28482 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL289139 0.84 KDM4E (0.86) KDM4EALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL288534 0.84 KDM4E (0.86) KDM4EALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL290132 0.83 KDM4E (1.00) KDM4EALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL289888 0.80 KDM4E (0.60) KDM4EALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL3827647 0.79 KDM4E (0.69) KDM4EALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL289147 0.78 KDM4E (0.67) KDM4EALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL290278 0.77 KDM4E (0.66) KDM4EALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL290099 0.77 KDM4E (0.81) KDM4EALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL289156 0.76 ALDH1A1 (0.65) KDM4EALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL289847 0.76 KDM4E (0.64) KDM4EALDH1A1RAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed