SCHEMBL29008185

SCHEMBL29008185

C=C(OCC)c1ccnc(C(=C)C)c1N

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
KMT2A Q03164 1/20 0.33
IKBKB O14920 1/20 0.32
BRD4 O60885 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TP53 P04637 1/20 0.30
HPGD P15428 1/20 0.30
CHEK2 O96017 1/20 0.30
NOS3 P29474 2/20 0.30
NOS2 P35228 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23234668 0.80 HRH4 (0.33) HRH4NOS3NOS2
SCHEMBL29663602 0.76 KDM4E (0.37) IKBKBALDH1A1
SCHEMBL17619234 0.76 KDM4E (0.37) IKBKBALDH1A1
SCHEMBL21608277 0.73 NOS2 (0.52) KMT2AHRH4NOS3NOS2
SCHEMBL23137481 0.72 PRKCI (0.35) IKBKBHRH4NOS3NOS2
SCHEMBL15758316 0.72 NUDT1 (0.51) NUDT1NPC1RAB9AKMT2ABRD4
SCHEMBL31522898 0.71 BRD4 (0.32) NPC1RAB9ABRD4ALDH1A1HSD17B10
SCHEMBL8296523 0.70 NAPRT (0.47) NPC1RAB9AALDH1A1HSD17B10TP53
SCHEMBL20509939 0.70 KDR (0.37) NUDT1NPC1RAB9AKMT2AALDH1A1
SCHEMBL21542765 0.70 NOS3 (0.38) KMT2AHRH4NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116171155-B Pyrido [2,3-d ] pyrimidine-2 (1H) -ketone derivative, preparation method and application thereof 上海和誉生物医药科技有限公司 2024-09-17 CN disclosed
CN-116171155-A Pyrido [2,3-d ] pyrimidine-2 (1H) -ketone derivative, preparation method and application thereof 上海和誉生物医药科技有限公司 2023-05-26 CN disclosed
WO-2022121839-A1 PYRIDO[2,3-D]PYRIMIDIN-2(1H)-ONE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 上海和誉生物医药科技有限公司 2022-06-16 WO disclosed