SCHEMBL29663602

SCHEMBL29663602

C=C(C)c1nccc(C(C)=O)c1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.37
ASPH Q12797 2/20 0.37
KDM8 Q8N371 2/20 0.37
PRKCI P41743 4/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
LIMK1 P53667 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
ATR Q13535 1/20 0.33
ALDH1A1 P00352 4/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
BLM P54132 1/20 0.32
AGER Q15109 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
IKBKB O14920 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17619234 1.00 KDM4E (0.37) KDM4EASPHKDM8PRKCIPDE3B
SCHEMBL23234668 0.87 HRH4 (0.33) KDM4EASPHKDM8
SCHEMBL21198627 0.84 KDM4E (0.38) KDM4EASPHKDM8PRKCIPDE3B
SCHEMBL17603745 0.83 KDM4E (0.47) KDM4EKDM4CATRALDH1A1MAPT
SCHEMBL30898769 0.77 NOS3 (0.48) PRKCILIMK1KDM4CATRALDH1A1
SCHEMBL23234804 0.77 PIK3C3 (0.37) KDM4EASPHKDM8PRKCIALDH1A1
SCHEMBL20520321 0.76 KDM4E (0.50) KDM4EASPHKDM8PDE3BPDE3A
SCHEMBL29008185 0.76 NUDT1 (0.34) ALDH1A1IKBKB
SCHEMBL21608277 0.76 NOS2 (0.52) KDM4ELIMK1
SCHEMBL30590435 0.76 SMN1; SMN2 (0.42) KDM4ELIMK1KDM4CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116171155-B Pyrido [2,3-d ] pyrimidine-2 (1H) -ketone derivative, preparation method and application thereof 上海和誉生物医药科技有限公司 2024-09-17 CN disclosed
CN-116171155-A Pyrido [2,3-d ] pyrimidine-2 (1H) -ketone derivative, preparation method and application thereof 上海和誉生物医药科技有限公司 2023-05-26 CN disclosed
WO-2022121839-A1 PYRIDO[2,3-D]PYRIMIDIN-2(1H)-ONE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 上海和誉生物医药科技有限公司 2022-06-16 WO disclosed