SCHEMBL29009559

SCHEMBL29009559

C=CS(=O)(=O)Nc1ccc2[nH]nc(-c3nc4ccccc4n3C3CNCCO3)c2c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.47
MAPK3 P27361 1/20 0.47
ITK Q08881 6/20 0.36
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
HRH1 P35367 1/20 0.34
KCNH2 Q12809 1/20 0.34
PDPK1 O15530 2/20 0.33
AURKA O14965 2/20 0.33
AURKB Q96GD4 1/20 0.33
TTK P33981 1/20 0.33
MET P08581 1/20 0.33
AXL P30530 3/20 0.32
MAPK10 P53779 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29009499 0.86 AURKA (0.42) ITKPDPK1AURKAAURKBMAPK10
SCHEMBL29009507 0.83 HRH1 (0.32) CYP3A4CYP2D6HRH1KCNH2
SCHEMBL29009516 0.76 EGFR (0.35) CYP3A4CYP2D6HRH1KCNH2AURKA
SCHEMBL29009558 0.72 MAPK3 (0.48) MAPK1MAPK3PDPK1
SCHEMBL29009534 0.71 HRH1 (0.37) CYP3A4CYP2D6HRH1KCNH2
SCHEMBL29009535 0.67 HRH1 (0.35) MAPK1CYP3A4CYP2D6HRH1KCNH2
SCHEMBL29009554 0.64 PDPK1 (0.66) PDPK1
SCHEMBL30382123 0.64 PDPK1 (0.66) PDPK1
SCHEMBL29009505 0.62 MAPK1 (0.59) MAPK1MAPK3ITKPDPK1
SCHEMBL29009498 0.60 FGFR1 (0.62) MAPK1MAPK3PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116217551-A Substituted indazole or azaindazole compounds and application thereof 河南中医药大学 2023-06-06 CN claimed
CN-116217551-A Substituted indazole or azaindazole compounds and application thereof 河南中医药大学 2023-06-06 CN disclosed